Hsp70 acts as a fine-switch that controls E3 ligase CHIP-mediated TAp63 and ΔNp63 ubiquitination and degradation

H Helena Wu1, Benfan Wang1, Stephen R Armstrong1

  • 1370 Heritage Medical Research Center, Department of Laboratory Medicine and Pathology, University of Alberta, Edmonton, Alberta T6G 2S2, Canada.

Nucleic Acids Research
|February 23, 2021
PubMed

Insights

Heat shock protein 70 (Hsp70) regulates cancer metastasis by controlling the degradation of p63 isoforms via the E3 ligase CHIP. This discovery reveals a new pathway for stabilizing p63 in cancers.

Area of Science:

  • Oncology
  • Molecular Biology
  • Cell Biology

Background:

  • Metastasis causes 90% of cancer deaths, with TAp63 suppressing tumors and ΔNp63 promoting them.
  • The precise mechanisms regulating p63 stability by ubiquitin E3 ligases are not fully understood.

Purpose of the Study:

  • To elucidate the role of CHIP (an E3 ligase) in p63 regulation.
  • To investigate the function of Hsp70 as a molecular switch in p63 degradation.
  • To determine how the Hsp70-CHIP axis impacts cancer cell migration and invasion.

Main Methods:

  • Investigated the interaction between CHIP and p63.
  • Utilized siRNA to deplete Hsp70 in cancer cell lines (H1299 and SCC9).
  • Assessed the impact of Hsp70 depletion on p63 isoform stability and interactions with CHIP.

Main Results:

  • CHIP directly interacts with p63 and promotes its degradation.
  • Hsp70 depletion stabilizes TAp63 and destabilizes ΔNp63, depending on the cell type.
  • Hsp70 modulates the interaction between p63 isoforms and CHIP, controlling ubiquitination and degradation.
  • The Hsp70-CHIP pathway influences tumor cell migration and invasion.

Conclusions:

  • Hsp70 acts as a molecular switch regulating CHIP-mediated ubiquitination and degradation of TAp63 and ΔNp63.
  • This identifies a novel pathway controlling p63 isoform stability in cancer.
  • Targeting the Hsp70-CHIP axis may offer new therapeutic strategies for managing cancer metastasis.

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