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Updated: Nov 15, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Allosteric Modulation of GPCRs of Class A by Cholesterol

Jan Jakubík1, Esam E El-Fakahany2

  • 1Department of Neurochemistry, Institute of Physiology Czech Academy of Sciences, 142 20 Prague, Czech Republic.

International Journal of Molecular Sciences
|March 6, 2021
PubMed

Keywords:
GPCRsallosteric modulationcholesterol

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