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Modulation of the Passive Permeability of Semipeptidic Macrocycles: N- and C-Methylations Fine-Tune Conformation and

Christian Comeau1, Benjamin Ries2, Thomas Stadelmann2

  • 1Département de Pharmacologie-Physiologie, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001, 12e av nord, Sherbrooke, Quebec, Canada J1H5N4.

Journal of Medicinal Chemistry
|March 22, 2021
PubMed

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