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Updated: Nov 10, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Emerging paradigms in activation, signaling, and regulation of G protein-coupled receptors

Arun K Shukla1

  • 1Department of Biological Sciences and Bioengineering, Indian Institute of Technology, Kanpur, India.

The FEBS Journal
|April 5, 2021
PubMed

Keywords:
GPCRsarrestinsbiased agonismcellular signalingdesensitization

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