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Updated: Nov 9, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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GPCRs that Rhoar the Guanine nucleotide exchange factors

Aishwarya Omble1,2, Kiran Kulkarni1,2

  • 1Division of Biochemical Sciences, CSIR-National Chemical Laboratory, Pune, India.

Small Gtpases
|April 14, 2021
PubMed

Keywords:
Cell migrationG protein-coupled receptors (GPCRs)Rho GTPasescell signallingexchange factors (GEFs)guanine nucleotide

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