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Functional Selectivity Does Not Predict Antinociceptive/Locomotor Impairing Potencies of NOP Receptor Agonists

Joaquim Azevedo Neto1, Chiara Ruzza1,2, Chiara Sturaro1

  • 1Section of Pharmacology, Department of Neuroscience and Rehabilitation, University of Ferrara, Ferrara, Italy.

Frontiers in Neuroscience
|April 16, 2021
PubMed

Keywords:
AT-403MCOPPBNOP receptorRo 65-6570functional selectivitymicenociceptin/orphanin FQβ arrestin 2 knockout mice

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