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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Discovery, optimization, and evaluation of non-bile acid FXR/TGR5 dual agonists

Sachiho Miyata1, Yuji Kawashima2, Miku Sakai3

  • 1Research Laboratory 1, FUJI YAKUHIN. CO., LTD, 1-32-3, Nishi-Omiya, Nishi-ku, Saitama City, Saitama, Japan. s-miyata@fujiyakuhin.co.jp.

Scientific Reports
|April 29, 2021
PubMed

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