Related Experiment Video

Updated: Nov 5, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Pharmacological selection of cannabinoid receptor effectors: Signalling, allosteric modulation and bias

Jamie J Manning1, Hayley M Green1, Michelle Glass1

  • 1Department of Pharmacology and Toxicology, University of Otago, Dunedin, New Zealand, PO Box 56, Dunedin, 9054, New Zealand.

Neuropharmacology
|May 17, 2021
PubMed

Keywords:
Allosteric modulationBiased agonismCannabinoid receptorFunctional selectivityG protein coupled receptorSignal transduction

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