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Mechanistic study of bergamottin-induced inactivation of CYP2C9

Ying Liu1, Shiyu Zhang1, Tingting Jiang1

  • 1State Key Laboratory of Functions and Applications of Medicinal Plants, Guizhou Provincial Key Laboratory of Pharmaceutics, Guizhou Medical University, Guiyang, 550004, Guizhou, PR China; School of Pharmacy, Guizhou College Medical University, Guiyang, 550004, Guizhou, PR China.

Food and Chemical Toxicology : an International Journal Published for the British Industrial Biological Research Association
|May 21, 2021
PubMed

Keywords:
BergamottinCYP2C9Drug-drug interactionGrapefruitMechanism-based inactivation

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