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"Clicking" fragment leads to novel dual-binding cholinesterase inhibitors

Zuzanna Molęda1, Anna Zawadzka1, Zbigniew Czarnocki1

  • 1University of Warsaw, Faculty of Chemistry, Pasteura 1, 02-093 Warsaw, Poland.

Bioorganic & Medicinal Chemistry
|June 15, 2021
PubMed

Keywords:
Combinatorial librariesGalantamineHybrid drugsStructure-activity relationshipTarget-guided synthesisTetrahydroisoquinolineTriazoleTryptamine”click” chemistry

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