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Activities of five new fluoroquinolones against Pseudomonas pseudomallei

M D Winton1, E D Everett, S A Dolan

  • 1Division of Infectious Diseases, University of Missouri-Columbia 65212.

Insights

This study tested five fluoroquinolones against Pseudomonas pseudomallei. Ciprofloxacin showed the most activity, but results suggest fluoroquinolones are not optimal for treating melioidosis.

Area of Science:

  • Microbiology
  • Infectious Diseases
  • Pharmacology

Background:

  • Melioidosis is a serious infectious disease caused by *Pseudomonas pseudomallei*.
  • Antimicrobial resistance is a growing concern in treating melioidosis.
  • Fluoroquinolones are a class of antibiotics with broad-spectrum activity.

Purpose of the Study:

  • To evaluate the in vitro susceptibility of *Pseudomonas pseudomallei* isolates to five fluoroquinolone antibiotics.
  • To determine the potential role of fluoroquinolones in melioidosis therapy.

Main Methods:

  • Broth microdilution technique was used.
  • Thirty-four clinical isolates of *Pseudomonas pseudomallei* were tested.
  • Susceptibility testing included amifloxacin, ciprofloxacin, enoxacin, norfloxacin, and ofloxacin.

Main Results:

  • Ciprofloxacin demonstrated the highest in vitro activity among the tested fluoroquinolones.
  • The minimum inhibitory concentration (MIC) for 90% of strains (MIC90) for ciprofloxacin was 8 µg/ml.
  • Other tested fluoroquinolones showed less activity.

Conclusions:

  • The in vitro activity of the tested fluoroquinolones against *Pseudomonas pseudomallei* suggests they may not be optimal for melioidosis treatment.
  • Further research into alternative or combination therapies is warranted.

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