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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Synthesis, bioevaluation and docking studies of new imidamide derivatives as nitric oxide synthase inhibitors

Fabio Arias1, Francisco Franco-Montalban1, Miguel Romero2

  • 1Departamento de Química Farmacéutica y Orgánica, Facultad de Farmacia, Universidad de Granada, Spain.

Bioorganic & Medicinal Chemistry
|July 4, 2021
PubMed

Keywords:
Drug designImidamidesInhibitorsNitric Oxide SynthaseSynthesis

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