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Opportunities and Challenges of Small Molecule Induced Targeted Protein Degradation

Ming He1, Wenxing Lv1, Yu Rao1

  • 1MOE Key Laboratory of Protein Sciences, School of Pharmaceutical Sciences, MOE Key Laboratory of Bioorganic Phosphorus Chemistry & Chemical Biology, Tsinghua University, Beijing, China.

Frontiers in Cell and Developmental Biology
|July 12, 2021
PubMed

Keywords:
E3 ubiquitin ligasePROTACproteasomeprotein degradationsmall molecule inhibitor

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