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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Discovery of tert-amine-based RORγt agonists

Ruomeng Qiu1, Mingcheng Yu1, Juwen Gong1

  • 1Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai, 201203, China.

European Journal of Medicinal Chemistry
|July 24, 2021
PubMed

Keywords:
Cancer immunotherapyRORγt agonistsSmall molecule drugsTertiary aminesTh17 cell differentiation

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