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Updated: Oct 15, 2025

A11-positive β-amyloid Oligomer Preparation and Assessment Using Dot Blotting Analysis
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Histamine H3 receptor antagonists with peptidomimetic (keto)piperazine structures to inhibit Aβ oligomerisation

Markus Falkenstein1, David Reiner-Link1, Aleksandra Zivkovic1

  • 1Institute of Pharmaceutical and Medicinal Chemistry, Heinrich Heine University Düsseldorf, Universitaetsstr. 1, 40225 Duesseldorf, Germany.

Bioorganic & Medicinal Chemistry
|October 25, 2021
PubMed

Keywords:
Alzheimeŕs diseaseHistamine H(3) receptorMulti target directed ligandsPeptidomimeticsProtein protein interactionβ-amyloid plaques

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