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Updated: Oct 15, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Structure-activity relationship study of hydroxyethylamine isostere and P1' site structure of peptide mimetic BACE1

Kazuya Kobayashi1, Takuya Otani1, Saki Ijiri1

  • 1Department of Medicinal Chemistry, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto 607-8412, Japan.

Bioorganic & Medicinal Chemistry
|October 26, 2021
PubMed

Keywords:
Alzheimer’s diseaseBACE1HydroxyethylamineInhibitorPeptide mimetics

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