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Closed-state inactivation and pore-blocker modulation mechanisms of human CaV2.2

Yanli Dong1, Yiwei Gao1, Shuai Xu2

  • 1National Laboratory of Biomacromolecules, CAS Center for Excellence in Biomacromolecules, Institute of Biophysics, Chinese Academy of Sciences, Beijing 100101, China; State Key Laboratory of Brain and Cognitive Science, Institute of Biophysics, Chinese Academy of Sciences, 15 Datun Road, Beijing 100101, China; College of Life Sciences, University of Chinese Academy of Sciences, Beijing 100049, China.

Cell Reports
|November 3, 2021
PubMed

Keywords:
Ca(V)2.2N-typechannel blockerclosed-state inactivationneurotransmitter releasepresynapsevoltage-gated calcium channelziconotide

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