Nanotherapeutics approaches to overcome P-glycoprotein-mediated multi-drug resistance in cancer
Jitu Halder1, Deepak Pradhan1, Biswakanth Kar1
1School of Pharmaceutical Science, Siksha 'O' Anusandhan (Deemed to be University), Bhubaneswar, Odisha, India.
Abstract:
Multidrug resistance (MDR) in cancer chemotherapy is a growing concern for medical practitioners. P-glycoprotein (P-gp) overexpression is one of the major reasons for multidrug resistance in cancer chemotherapy. The P-gp overexpression in cancer cells depends on several factors like adenosine triphosphate (ATP) hydrolysis, hypoxia-inducible factor 1 alpha (HIF-1α), and drug physicochemical properties such as lipophilicity, molecular weight, and molecular size. Further multiple exposures of anticancer drugs to the P-gp efflux protein cause acquired P-gp overexpression. Unique structural and functional characteristics of nanotechnology-based drug delivery systems provide opportunities to circumvent P-gp mediated MDR. The primary mechanism behind the nanocarrier systems in P-gp inhibition includes: bypassing or inhibiting the P-gp efflux pump to combat MDR. In this review, we discuss the role of P-gp in MDR and highlight the recent progress in different nanocarriers to overcome P-gp mediated MDR in terms of their limitations and potentials.
Insights
Multidrug resistance (MDR) in cancer is often caused by P-glycoprotein (P-gp) overexpression. Nanotechnology offers promising strategies to bypass or inhibit P-gp efflux pumps, overcoming chemotherapy resistance.
Area of Science:
- Oncology
- Nanotechnology
- Pharmacology
Background:
- Multidrug resistance (MDR) is a significant challenge in cancer chemotherapy.
- P-glycoprotein (P-gp) overexpression is a primary driver of MDR, influenced by factors like ATP hydrolysis and drug properties.
Purpose of the Study:
- To review the role of P-gp in MDR.
- To highlight recent advancements in nanocarrier systems for overcoming P-gp mediated MDR.
Main Methods:
- Discussion of P-gp overexpression mechanisms.
- Review of nanotechnology-based drug delivery systems.
- Analysis of nanocarrier limitations and potentials.
Main Results:
- P-gp overexpression is linked to ATP hydrolysis, HIF-1α, and drug physicochemical properties.
- Nanocarriers can bypass or inhibit P-gp efflux pumps.
- Various nanocarrier systems show potential in combating MDR.
Conclusions:
- Nanotechnology-based systems offer unique advantages to circumvent P-gp mediated MDR.
- Further research into nanocarrier limitations and potentials is crucial for clinical application.
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