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Updated: Oct 12, 2025

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Tandem Amination/Oxetane Ring Opening toward Benzomorpholines

Lindsey G DeRatt1, Chao-Yuan Wang1, Scott D Kuduk1

  • 1Janssen Research and Development, 1400 McKean Road, Spring House, Pennsylvania 19477, United States.

The Journal of Organic Chemistry
|November 22, 2021
PubMed

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