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Updated: Oct 12, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

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Targeting cyclin-dependent kinase 9 in cancer therapy

Yi-Li Shen1, Yan-Mao Wang1, Ya-Xin Zhang1

  • 1Division of Pulmonary Medicine, The First Affiliated Hospital of Wenzhou Medical University, Key Laboratory of Heart and Lung, Wenzhou, 325000, China.

Acta Pharmacologica Sinica
|November 23, 2021
PubMed

Keywords:
CDK9CDK9 inhibitorscancerepigenetic regulationtranscription

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