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Updated: Oct 11, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Neurosteroid Modulation of GABAA Receptor Function by Independent Action at Multiple Specific Binding Sites

Lei Wang1,2, Douglas F Covey1,3,4, Gustav Akk1,5

  • 1Department of Anesthesiology (LW, DFC, GA, ASE),Union Hospital, Tongji Medical College, Huazhong University of Science and Technology, Wuhan, Hubei , China.

Current Neuropharmacology
|December 3, 2021
PubMed

Keywords:
GABANeurosteroidsaffinity labelingdesensitizationion channelsstructural biology

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