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Updated: Oct 8, 2025

A Practical Guide for the Production and PET/CT Imaging of 68Ga-DOTATATE for Neuroendocrine Tumors in Daily Clinical Practice
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Distinct In Vitro Binding Profile of the Somatostatin Receptor Subtype 2 Antagonist [177Lu]Lu-OPS201 Compared to the

Rosalba Mansi1, Pascale Plas2, Georges Vauquelin3

  • 1Division of Radiopharmaceutical Chemistry, Clinic of Radiology and Nuclear Medicine, University Hospital Basel, University of Basel, 4031 Basel, Switzerland.

Pharmaceuticals (Basel, Switzerland)
|December 28, 2021
PubMed

Keywords:
[177Lu]Lu-DOTA-TATE[177Lu]Lu-OPS201binding sitesdissociationkineticsradioligand bindingsomatostatin receptor

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