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Molecular Design, Synthesis, and Evaluation of SNIPER (ER) that Induces Targeted Protein Degradation of ERα

Nobumichi Ohoka1, Hidetomo Yokoo2, Keiichiro Okuhira1,3

  • 1Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences, Kawasaki, Kanagawa, Japan.

Methods in Molecular Biology (Clifton, N.J.)
|February 4, 2022
PubMed

Keywords:
Antitumor activityCell deathEstrogen receptorProtein knockdownSNIPERUbiquitin-proteasome system

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