Related Experiment Video

Updated: Oct 2, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Ligands and Beyond: Mechanosensitive Adhesion GPCRs

Hsi-Hsien Lin1,2,3, Kwai-Fong Ng2, Tse-Ching Chen2

  • 1Department of Microbiology and Immunology, College of Medicine, Chang Gung University, Taoyuan 33302, Taiwan.

Pharmaceuticals (Basel, Switzerland)
|February 26, 2022
PubMed

Keywords:
GPCR activationGPS autoproteolysisadhesion GPCRmechanotransductionsignalingtethered ligand

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