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Focus on the classical and non-classical functions of EZH2: Guide the development of inhibitors and degraders

Qiangsheng Zhang1, Hongling Yang1, Qiang Feng2

  • 1State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, West China Medical School, Sichuan University, and Collaborative Innovation Center for Biotherapy, 17#3rd Section, Ren Min South Road, Chengdu 610041, China.

Pharmacological Research
|March 8, 2022
PubMed

Keywords:
Covalent inhibitorsDegradersDual inhibitorsEZH2EpigeneticsHistone modificationPPI inhibitors

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