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Cyclobutanes in Small-Molecule Drug Candidates

Marnix R van der Kolk1, Mathilde A C H Janssen1, Floris P J T Rutjes1

  • 1Institute for Molecules and Materials, Radboud University, Heyendaalseweg 135, 6526 AJ, Nijmegen, The Netherlands.

Chemmedchem
|March 9, 2022
PubMed

Keywords:
Cyclobutanesconformational restrictionisosterespharmacophoresstrained carbocycles

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