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Updated: Sep 30, 2025

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
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Anthraquinone derivatives as ADP-competitive inhibitors of liver pyruvate kinase

Amalyn Nain-Perez1, Anders Foller Füchtbauer1, Liliana Håversen2

  • 1Department of Chemistry and Molecular Biology, University of Gothenburg, SE-412 96, Gothenburg, Sweden.

European Journal of Medicinal Chemistry
|March 15, 2022
PubMed

Keywords:
ADP competitive inhibitorsEnzymatic inhibitionLiver pyruvate kinaseNon-alcoholic fatty liver diseaseStructure-activity relationship

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