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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Chemical Synthesis, Pharmacokinetic Properties and Biological Effects of JM-00266, a Putative Non-Brain Penetrant

Tania Muller1, Laurent Demizieux1, Stéphanie Troy-Fioramonti1

  • 1Equipe Physiopathologie des dyslipidémies, Unité Mixte de Recherche Université de Bourgogne Franche-Comté - Institut National de la Santé et de la Recherche Médicale (UMR-INSERM) 1231, F-21000 Dijon, France.

International Journal of Molecular Sciences
|March 25, 2022
PubMed

Keywords:
CB1R antagonistRimonabantSWISSADME predictiondrug discoveryendocannabinoid systemobesitypharmacokinetics

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