Recent Progress of Bioactivities, Mechanisms of Action, Total Synthesis, Structural Modifications and

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Updated: Sep 28, 2025

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

8.3K

Tianze Li1, Hui Xu1,2

  • 1College of Plant Protection, Northwest A&F University, Yangling 712100, Shaanxi Province, P.R. China.

Mini Reviews in Medicinal Chemistry
|April 1, 2022
PubMed

Keywords:
Indolebiological activityindole derivativesmechanism of actionstructural modificationstructural- activity relationshiptotal synthesis

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