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Updated: Sep 27, 2025

Synthesis and Characterization of Functionalized Metal-organic Frameworks
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Adjusted degradation of BRD4 S and BRD4 L based on fine structural modifications of the pyrrolopyridone scaffold

Jingjing Chen1, Huixin He2, Aihuan Wei3

  • 1School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, UCAS, 1 Xiangshanzhi Road, Hangzhou, 310024, China.

European Journal of Medicinal Chemistry
|April 8, 2022
PubMed

Keywords:
BRD4 SPROTACPyrrolopyridoneSelectivity

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