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Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor

Jigar Desai1, Bhaumin Patel1, Archana Gite1

  • 1Zydus Research Centre, Cadila Healthcare Ltd, Sarkhej-Bavla N.H. No. 8A, Moraiya, Ahmedabad 382210, India.

Bioorganic & Medicinal Chemistry Letters
|April 12, 2022
PubMed

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Keywords:
InflammationJAK inhibitorMomelotinibPyrimidine