Antiplatelet response to clopidogrel is associated with a haplotype in CYP2C19 gene in Pakistani patients

Sagheer Ahmed1, Saima Gul2, Sami Siraj3

  • 1Shifa College of Pharmaceutical Sciences, Shifa Tameer-e-Millat University, Islamabad, Pakistan.

Scientific Reports
|April 14, 2022
PubMed

Insights

Clopidogrel response varies, with CYP2C19*2 allele common in Pakistan. Haplotype, blood glucose, and diabetes history, not just genotype, impact clopidogrel effectiveness in preventing ischemic events.

Area of Science:

  • Pharmacogenomics
  • Cardiovascular Medicine
  • Clinical Chemistry

Background:

  • Clopidogrel is a vital antiplatelet medication for ischemic diseases.
  • Poor platelet inhibition can lead to treatment failure despite clopidogrel use.
  • CYP2C19 genetic variations influence clopidogrel metabolism and efficacy.

Purpose of the Study:

  • To examine the association of CYP2C19 polymorphisms and clinical factors with clopidogrel's antiplatelet response in a Pakistani cohort.
  • To identify predictors of clopidogrel resistance in patients with cardiovascular diseases.

Main Methods:

  • Genotyping for CYP2C19*2 and *3 alleles in 120 cardiovascular patients on clopidogrel.
  • Monitoring antiplatelet response using Helena AggRAM, categorizing patients into high and low responders.
  • Analyzing associations between genetic variations, clinical data (leukocyte count, blood glucose, diabetes history), and response phenotypes.

Main Results:

  • CYP2C19*2 allele prevalence was 38.3% (one copy) and 5% (two copies); no *3 allele detected.
  • No significant difference in response based on CYP2C19 metabolizer status (extensive, intermediate, poor).
  • Haplotype H1, leukocyte count, random blood glucose, and diabetes history were significantly associated with clopidogrel response.

Conclusions:

  • CYP2C19 genotype alone does not fully predict clopidogrel response in this Pakistani cohort.
  • Clinical factors like blood glucose and diabetes history are important determinants of clopidogrel efficacy.
  • Findings highlight the need for personalized antiplatelet therapy considering genetic and clinical variables.

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