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Updated: Sep 27, 2025

Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay
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Parallel Interrogation of β-Arrestin2 Recruitment for Ligand Screening on a GPCR-Wide Scale using PRESTO-Tango Assay

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Ligand-based pharmacophore modeling, virtual screening and biological evaluation to identify novel TGR5 agonists

Shizhen Zhao1, Xinping Li1, Wenjing Peng1

  • 1Key Laboratory of Receptors-Mediated Gene Regulation and Drug Discovery, People's Hospital of Hebi, School of Medicine, Henan University Henan China hb_lwg@163.com.

RSC Advances
|April 15, 2022
PubMed

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