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Development of novel androgen receptor antagonists based on the structure of darolutamide

Qian Xu1, Zixiong Zhang2, Chenchao Huang1

  • 1Key Laboratory of the Ministry of Education for Advanced Catalysis Materials, Department of Chemistry, Zhejiang Normal University, 688 Yingbin Road, Jinhua 321004, China.

Bioorganic Chemistry
|May 1, 2022
PubMed

Keywords:
Androgen receptor antagonistCRPCDarolutamideStructure-activity relationship

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