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Advances and perspectives of proteolysis targeting chimeras (PROTACs) in drug discovery

Jia-Yue Xi1, Ru-Yue Zhang1, Ke Chen1

  • 1Department of Pharmaceutical Chemistry and Analysis, Fourth Military Medical University, Xi'an, Shaanxi 710032, China.

Bioorganic Chemistry
|May 9, 2022
PubMed

Keywords:
Drug discoveryPROTACsSmall inhibitorsTarget protein degradationUndruggable target

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