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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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An efficient route to N-alkylated 3,4-dihydroisoquinolinones with substituents at the 3-position

Aoi Tazawa1,2, Junki Ando1, Kohei Ishizawa1

  • 1Sohyaku Innovative Research Division, Mitsubishi Tanabe Pharma Corporation 1000 Kamoshida-cho, Aoba-ku Yokohama-shi Kanagawa 227-0033 Japan tanaka.minoru@mw.mt-pharma.co.jp.

RSC Advances
|May 11, 2022
PubMed

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