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Updated: Sep 21, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

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Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with

Martin Juhás1, Andrea Bachtíková1, Daria Elżbieta Nawrot1

  • 1Faculty of Pharmacy in Hradec Králové, Charles University, Akademika Heyrovského 1203, 500 05 Hradec Králové, Czech Republic.

Pharmaceuticals (Basel, Switzerland)
|May 28, 2022
PubMed

Keywords:
aminooxazoleaminothiazoleantimycobacterial activitydockingisosteremolecular dockingmolecular dynamicspyridinewater solubility

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