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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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2-Arylindoles: Concise Syntheses and a Privileged Scaffold for Fungicide Discovery

Jingqian Huo1, Lai Chen1, Helong Si1

  • 1College of Plant Protection, Hebei Agricultural University, Baoding 071001, P. R. China.

Journal of Agricultural and Food Chemistry
|June 6, 2022
PubMed

Keywords:
2-arylindole derivativesfungicidal activityone-pot synthesis

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