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Updated: Sep 20, 2025

Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs
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Biphenyl Ether Analogs Containing Pomalidomide as Small-Molecule Inhibitors of the Programmed Cell Death-1/Programmed

Shabnam Shaabani1, Louis Gadina2, Ewa Surmiak2

  • 1Department of Drug Design, University of Groningen, 9713 AV Groningen, The Netherlands.

Molecules (Basel, Switzerland)
|June 10, 2022
PubMed

Keywords:
PD-1/PD-L1immune checkpoint blockadesmall-molecule inhibitors

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