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Updated: Sep 20, 2025

Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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Superacid-Mediated Late-Stage Aromatic Polydeuteration of Pharmaceuticals

Emeline Appert1,2, Agnès Martin-Mingot1, Omar Karam2

  • 1Superacid Group - Organic Synthesis Team, IC2MP, Université de Poitiers, UMR-CNRS 7285, 4 rue Michel Brunet, TSA 51106, 86073, Poitiers Cedex 9, France.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|June 11, 2022
PubMed

Keywords:
alkaloidsdeuteriumisotope labelinglate-stage functionalizationsuperacid

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