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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Recent Progress in the Synthesis of Drugs and Bioactive Molecules Incorporating Nitro(het)arene Core

Maxim Bastrakov1, Alexey Starosotnikov1

  • 1N.D. Zelinsky Institute of Organic Chemistry RAS, Leninsky Prosp. 47, Moscow 19991, Russia.

Pharmaceuticals (Basel, Switzerland)
|June 24, 2022
PubMed

Keywords:
arenesbiological activitydrugsheterocyclesnitro group

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