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Updated: Sep 3, 2025

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay
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Discovery of two novel (4-hydroxyphenyl) substituted polycyclic carbocycles as potent and selective estrogen receptor

Edward A Wetzel1, Kylee J Marks2, Alexandra A Gleason2

  • 1Department of Chemistry, Marquette University, P. O. Box 1881, Milwaukee, WI 53201-1881, United States.

Bioorganic & Medicinal Chemistry Letters
|July 23, 2022
PubMed

Keywords:
DockingDrug developmentEstrogen receptor agonistSERBA

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