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Catalytic covalent inhibition of cyclooxygenase-1 by a biomimetic acyltransferase

Wei Bao1, Baruch Turniansky1, John Koh1

  • 1University of Delaware, 102 Brown Laboratory, Newark, DE 19716, USA.

Bioorganic & Medicinal Chemistry
|September 5, 2022
PubMed

Keywords:
Acyl-transfer catalysisCatalytic covalent inhibitorCovalent inhibitorCyclooxygenaseProtein acetylation

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