Losartan ameliorates renal interstitial fibrosis through metabolic pathway and Smurfs-TGF-β/Smad

Junju Zou1, Xiaotao Zhou2, Yuerong Ma2

  • 1Hunan Provincial Key Laboratory of Translational Research in TCM Prescriptions and Zheng, Hunan University of Chinese Medicine, Changsha, Hunan 410208, China.

Insights

Losartan treatment reduced renal fibrosis in mice with kidney injury. It improved renal function and inhibited key fibrotic pathways by promoting protein degradation via ubiquitination.

Area of Science:

  • Nephrology
  • Molecular Biology
  • Metabolomics

Background:

  • Renal fibrosis, a common endpoint for chronic kidney diseases, is driven by complex pathways including inflammation, oxidative stress, and metabolic dysfunction.
  • Epithelial-mesenchymal transition (EMT) in renal tubular cells is a critical mechanism underlying renal fibrosis.
  • Losartan, an Angiotensin II (ANG II) receptor antagonist, is known for its vasodilatory effects.

Purpose of the Study:

  • To investigate the therapeutic effects of losartan on renal fibrosis in a mouse model of Unilateral Ureteral Obstruction (UUO).
  • To explore the impact of losartan on the transforming growth factor-beta (TGF-β)/Smad signaling pathway and metabolomic profiles in the context of renal fibrosis.

Main Methods:

  • Establishment of a UUO model in male C57BL/6J mice.
  • Administration of losartan at doses of 10, 20, and 30 mg/kg/d for 28 consecutive days.
  • Analysis of serum metabolic spectrum, renal function, histological changes (tubulointerstitial injury, collagen deposition), and molecular markers (Smurf2, Smurf1, TβR-I, P-Smad2/3) related to TGF-β/Smad signaling and EMT.

Main Results:

  • Losartan treatment significantly ameliorated UUO-induced abnormalities in serum metabolic profiles and improved overall renal function.
  • Histological analysis revealed that losartan reduced tubulointerstitial dilation and collagen deposition, thereby mitigating renal tubular-interstitial injury and fibrosis.
  • Losartan promoted the nuclear expression of Smurf2 and Smurf1, E3 ubiquitin ligases, leading to the degradation of TGF-β1 type I receptor (TβR-I) and phosphorylated Smad2/3 (P-Smad2/3), consequently inhibiting renal tubular epithelial cell EMT.

Conclusions:

  • Losartan effectively reduces renal fibrosis in a mouse UUO model.
  • The antifibrotic effects of losartan are mediated through the regulation of the TGF-β/Smad pathway and metabolic alterations via ubiquitination.
  • Losartan demonstrates potential as a therapeutic agent for mitigating renal fibrosis by targeting EMT and associated molecular pathways.

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