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Paradoxical Increase of Permeability and Lipophilicity with the Increasing Topological Polar Surface Area within a

Upendra Argikar1, Markus Blatter2, Dallas Bednarczyk1

  • 1Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.

Journal of Medicinal Chemistry
|September 7, 2022
PubMed

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