Human islet amyloid polypeptide: A therapeutic target for the management of type 2 diabetes mellitus

Pratiksha H Roham1, Shreyada N Save1, Shilpy Sharma1

  • 1Department of Biotechnology, Savitribai Phule Pune University, Ganeshkhind, 41100, India.

Insights

Human islet amyloid polypeptide (hIAPP) aggregation contributes to pancreatic beta-cell loss in type 2 diabetes. Targeting hIAPP aggregation intermediates offers a promising therapeutic strategy for managing type 2 diabetes mellitus (T2DM).

Area of Science:

  • Biochemistry
  • Endocrinology
  • Molecular Biology

Background:

  • Type 2 diabetes mellitus (T2DM) lacks effective diagnostic markers, and current treatments only delay progression.
  • Misfolding and aggregation of human islet amyloid polypeptide (hIAPP) correlate with pancreatic beta-cell decline in T2DM.
  • hIAPP is a recognized therapeutic target for T2DM management.

Purpose of the Study:

  • To review hIAPP's role in pancreatic beta-cell dysfunction and apoptosis.
  • To explore hIAPP aggregation intermediates as potential drug targets for T2DM.
  • To discuss therapeutic agents that inhibit or reverse hIAPP aggregation.

Main Methods:

  • Literature review of hIAPP aggregation mechanisms in T2DM.
  • Analysis of hIAPP's role in endoplasmic reticulum stress, oxidative stress, and mitochondrial dysfunction.
  • Survey of therapeutic strategies targeting hIAPP aggregation.

Main Results:

  • hIAPP aggregation induces beta-cell apoptosis through various cellular stresses and autophagy blockade.
  • hIAPP aggregation intermediates present viable targets for T2DM drug development.
  • Diverse agents, including small molecules, natural compounds, and nanoparticles, show potential in inhibiting hIAPP aggregation.

Conclusions:

  • hIAPP aggregation is a key factor in T2DM pathogenesis.
  • Targeting hIAPP aggregation pathways offers a novel therapeutic avenue for T2DM.
  • Further development of hIAPP aggregation inhibitors could lead to disease-modifying therapies for T2DM.

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