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Construction of Cyclic Cell-Penetrating Peptides for Enhanced Penetration of Biological Barriers
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Inhibitory prodrug mechanism for cysteine cathepsin-targeted self-controlled drug release

Floris J van Dalen1, Martijn Verdoes1

  • 1Department of Tumour Immunology and the Institute for Chemical Immunology, Radboud Institute for Molecular Life Sciences, Radboud University Medical Centre, Nijmegen, Netherlands.

Journal of Enzyme Inhibition and Medicinal Chemistry
|September 19, 2022
PubMed

Keywords:
Inhibitory prodrugcysteine cathepsinsselective drug deliverytumour microenvironmenttumour-associated macrophages

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