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Discovery and Structural Explorations of G-Protein Biased μ-Opioid Receptor Agonists

Xiang Li1,2, Yanhao Guo3, Jing Li1

  • 1State Key Laboratory of Toxicology and Medical Countermeasures, Beijing Institute of Pharmacology & Toxicology, Beijing, 100850, P. R. China.

Chemmedchem
|October 9, 2022
PubMed

Keywords:
G-protein biased agonistsPZM21antinociceptiveβ-arrestin2 recruitmentμOR

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