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Updated: Aug 20, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Discovery of Potent Inhibitors of Cyclin-Dependent Kinases 7 and 9: Design, Synthesis, Structure-Activity

Renjie Chen1, Ramin Hassankhani1, Yi Long1

  • 1Drug Discovery and Development, Clinical and Health Sciences, University of South Australia, Adelaide, SA, 5000, Australia.

Chemmedchem
|November 18, 2022
PubMed

Keywords:
CDK7CDK9N-pyridinylpyrimidin-2-aminesinhibitorsstructure-activity relationships

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