Eukaryotic Transcription Activators
tRNA Activation
RNA Polymerase II Accessory Proteins
Epigenetic Regulation
Translesion DNA Polymerases
Abnormal Proliferation
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Updated: Aug 20, 2025

Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors
Published on: August 5, 2022
Amika Kikuchi1, Hiroki Onoda1,2, Kosuke Yamaguchi3
1Structural Biology Laboratory, Graduate School of Medical Life Science, Yokohama City University, Tsurumi-ku, Yokohama, Kanagawa, 230-0045, Japan.
Researchers uncovered how DNA methyltransferase 1 (DNMT1) is activated. A key linker region repositions domains, enabling DNMT1 to maintain DNA methylation, crucial for genomic stability and drug design.
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